SCHEMBL8208746

SCHEMBL8208746

Nc1nc2nc[nH]c2c(=O)n1Cc1ccc(-c2ccccc2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.45
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ADORA3 P0DMS8 4/20 0.39
ADORA2B P29275 2/20 0.39
CYP2E1 P05181 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
PDE4A P27815 5/20 0.39
PDE4B Q07343 5/20 0.39
PDE4C Q08493 5/20 0.39
PDE4D Q08499 5/20 0.39
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
CDK2 P24941 1/20 0.38
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208739 0.82 PNP (0.40) PNPCYP11B1CYP11B2CYP2E1CYP3A4
SCHEMBL3300188 0.81 PNP (0.40) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL4963422 0.81 PNP (0.40) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL9434524 0.81 PNP (0.40) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL18250 0.81 PNP (0.66) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL1980960 0.80 PNP (0.64) PNPADORA3ADORA2BPDE4APDE4B
SCHEMBL4962859 0.79 PDE4A (0.53) PNPADORA3ADORA2BCYP3A4CYP2C19
Hydrochloric Acid SCHEMBL18605981 0.78 PDE4A (0.53) PNPADORA3ADORA2BCYP3A4CYP2C19
SCHEMBL1938290 0.76 KMT2A (0.49) PNPADORA3ADORA2BCYP3A4CYP2C9
SCHEMBL9434882 0.76 PIN1 (0.52) PNPADORA3ADORA2BCYP2C19PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096724-A O(6)-ALKYLGUANINE-DNA ALKYLTRANSFERASE (ATASE) ENZYME INHIBITORS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-08-01 US disclosed