SCHEMBL4964950

SCHEMBL4964950

CCc1c(-c2ccccc2)sc(N)c1C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
MAPT P10636 5/20 0.57
GAA P10253 4/20 0.57
MEN1 O00255 1/20 0.57
LMNA P02545 1/20 0.57
KMT2A Q03164 1/20 0.57
GRM6 O15303 9/20 0.55
HPGD P15428 5/20 0.55
NPSR1 Q6W5P4 2/20 0.55
GRM5 P41594 1/20 0.50
ALOX15 P16050 3/20 0.47
HSD17B10 Q99714 3/20 0.47
USP2 O75604 1/20 0.47
RECQL P46063 1/20 0.47
TDP1 Q9NUW8 1/20 0.45
KDM4E B2RXH2 1/20 0.43
CASP1 P29466 1/20 0.43
IKBKB O14920 1/20 0.42
ADORA1 P30542 1/20 0.42
TP53 P04637 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10713203 0.89 ALDH1A1 (0.71) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL10714409 0.84 GRM6 (0.68) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL10713913 0.83 GRM6 (0.76) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL1382025 0.80 SMN1; SMN2 (0.48) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL4099130 0.80 GRM6 (0.74) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL20665498 0.78 GRM6 (0.62) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL1929543 0.77 GRM6 (0.70) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL4561915 0.76 ALDH1A1 (0.49) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL4093308 0.73 GRM6 (0.49) ALDH1A1MAPTGAAMEN1LMNA
SCHEMBL3452499 0.72 CYP1A2 (0.55) ALDH1A1MAPTGAAMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436279-B1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-08-13 EP claimed
EP-1436279-B1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-08-13 EP disclosed