SCHEMBL4965375

SCHEMBL4965375

CC(C)(C)c1ccccc1C(=O)N(c1ccc(O)cc1)c1ccc(OCCN2CCCCC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.67
ESR2 Q92731 4/20 0.67
PSMB1 P20618 3/20 0.48
PSMB5 P28074 3/20 0.48
PSMB2 P49721 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
HSD17B10 Q99714 1/20 0.48
HTT P42858 1/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
LTA4H P09960 1/20 0.47
ESRRG P62508 2/20 0.46
GCGR P47871 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788627 0.87 ESR1 (0.64) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL2113321 0.83 ESR1 (0.60) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL2111310 0.83 GCGR (0.64) ESR1ESR2HTTLTA4HGCGR
SCHEMBL2115656 0.82 LTA4H (0.62) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL2113940 0.82 KDM4E (0.61) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL10116921 0.81 ESR1 (0.82) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL2112716 0.81 LTA4H (0.64) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL2112820 0.81 ESR1 (0.64) ESR1ESR2PSMB1PSMB5PSMB2
Hydrochloric Acid SCHEMBL2115234 0.81 ESR1 (0.60) ESR1ESR2PSMB1PSMB5PSMB2
SCHEMBL10116793 0.80 ESR1 (1.00) ESR1ESR2PSMB1PSMB5PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954670-A2 NUCLEAR RECEPTOR BINDING AGENTS GTX Inc. (US) 2008-08-13 EP disclosed
WO-2007062230-A2 NUCLEAR RECEPTOR BINDING AGENTS GTX, INC. (US) 2007-05-31 WO disclosed