SCHEMBL4965526

SCHEMBL4965526

NC(=O)OCC(c1ccccc1Cl)n1nnnc1-c1cccc(Cl)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 12/20 0.44
TRPA1 O75762 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
KMT2A Q03164 1/20 0.35
CTSA P10619 1/20 0.35
ALDH1A1 P00352 1/20 0.34
KCNN4 O15554 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
AVPR2 P30518 1/20 0.34
AVPR1A P37288 1/20 0.34
NPBWR1 P48145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958219 0.79 MAPT (0.41) P2RX7MAPTTHRBKMT2ACTSA
SCHEMBL4310574 0.75 P2RX7 (0.52) P2RX7TRPA1SIGMAR1SLC6A2SLC6A4
SCHEMBL4962394 0.73 CYP2D6 (0.38) MAPTTHRBKMT2ACTSAALDH1A1
SCHEMBL4959671 0.71 CYP1A2 (0.37) MAPTTHRBCTSAALDH1A1AVPR2
SCHEMBL25345950 0.70 POLB (0.41) MAPTKMT2AALDH1A1SLC6A2SLC6A4
SCHEMBL4960190 0.70 POLB (0.41) MAPTKMT2AALDH1A1SLC6A2SLC6A4
SCHEMBL4957454 0.69 SMN1; SMN2 (0.41) MAPTTHRBKMT2AALDH1A1
SCHEMBL4311872 0.67 P2RX7 (0.49) P2RX7TRPA1SIGMAR1KMT2ACTSA
SCHEMBL4958417 0.67 MAPT (0.43) MAPTTHRBKMT2ACTSAALDH1A1
SCHEMBL3447381 0.66 CYP1A2 (0.46) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879873-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK Holdings Co., Ltd. (KR) 2008-01-23 EP disclosed
WO-2006112685-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK HOLDINGS CO., LTD. (KR) 2006-10-26 WO disclosed