SCHEMBL4965902

SCHEMBL4965902

CCc1ccc(C(=O)c2ccc(OC3CCC3)cc2Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
PARP10 Q53GL7 1/20 0.44
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
RORC P51449 1/20 0.39
SLC22A12 Q96S37 1/20 0.39
HIF1A Q16665 1/20 0.38
CNR2 P34972 2/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967870 0.85 PDE4D (0.45) ADRB2KMT2AMEN1PDE4APDE4B
SCHEMBL4967860 0.85 PDE4D (0.45) ADRB2KMT2AMEN1PDE4APDE4B
SCHEMBL14116655 0.85 PDE4D (0.45) ADRB2KMT2AMEN1PDE4APDE4B
SCHEMBL1252259 0.82 NPC1 (0.55) KMT2AMEN1MAPTHTTSMN1; SMN2
SCHEMBL4969314 0.81 POLB (0.39) ADRB2KMT2AMEN1MAPTHTT
SCHEMBL4968823 0.80 MAPT (0.51) KMT2AMEN1PARP10MAPTHTT
SCHEMBL4969219 0.79 MAPT (0.45) KMT2APARP10MAPTHTTSMN1; SMN2
SCHEMBL26121415 0.78 HIF1A (0.46) KMT2APARP10MAOAMAOBHIF1A
SCHEMBL8318438 0.76 MAOB (0.50) KMT2APARP10PDE4APDE4BPDE4C
SCHEMBL4969129 0.75 PDE5A (0.41) KMT2AMEN1MAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed