SCHEMBL4969314

SCHEMBL4969314

CCc1ccc(C(=O)c2cc(I)c(OC3CCC3)cc2Br)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
PDE5A O76074 2/20 0.39
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 3/20 0.37
ADRB2 P07550 2/20 0.37
MEN1 O00255 2/20 0.37
PDE4A P27815 4/20 0.36
PDE4B Q07343 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967088 0.86 PDE4D (0.45) PDE4APDE4BPDE4CPDE4D
SCHEMBL4966844 0.86 PDE4D (0.45) PDE4APDE4BPDE4CPDE4D
SCHEMBL1253373 0.82 MAPT (0.44) MAPTHTTSMN1; SMN2KMT2AMEN1
SCHEMBL4967215 0.81 HSD17B10 (0.47) MAPTHTTSMN1; SMN2KMT2AMEN1
SCHEMBL4966210 0.81 KMT2A (0.41) POLBMAPTKMT2AMEN1
SCHEMBL4965902 0.81 ADRB2 (0.46) MAPTHTTSMN1; SMN2KMT2AADRB2
SCHEMBL4968303 0.79 MAPT (0.41) MAPTHTTSMN1; SMN2KMT2AMEN1
SCHEMBL4969129 0.77 PDE5A (0.41) POLBPDE5AMAPTHTTSMN1; SMN2
SCHEMBL1252278 0.76 MAPT (0.47) POLBMAPTHTTSMN1; SMN2KMT2A
SCHEMBL4969708 0.75 MAPT (0.44) POLBMAPTHTTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed