SCHEMBL4967174

SCHEMBL4967174

CC(C#N)Cc1c[c]ccc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.34
TSHR P16473 1/20 0.33
SLC6A2 P23975 3/20 0.31
TAAR1 Q96RJ0 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
MAOA P21397 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
CYP2A6 P11509 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
HTR2A P28223 1/20 0.31
ADRA1A P35348 1/20 0.31
OPRK1 P41145 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL128086 0.80 TAAR1 (0.35) TSHRSLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL27932397 0.79 TAAR1 (0.34) TSHRSLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL9330630 0.79 TAAR1 (0.34) TSHRSLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL13593628 0.78 SIGMAR1 (0.52) MAOBTSHRSLC6A2TAAR1SLC6A4
SCHEMBL14452762 0.78 SIGMAR1 (0.52) MAOBTSHRSLC6A2TAAR1SLC6A4
SCHEMBL1752148 0.78 SIGMAR1 (0.52) MAOBTSHRSLC6A2TAAR1SLC6A4
SCHEMBL28049245 0.78
SCHEMBL3616684 0.77 TAAR1 (0.33) SLC6A2TAAR1SLC6A4SLC6A3MAOA
SCHEMBL3608914 0.77 TAAR1 (0.33) SLC6A2TAAR1SLC6A4SLC6A3MAOA
SCHEMBL3603367 0.77 TAAR1 (0.33) SLC6A2TAAR1SLC6A4SLC6A3MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966174-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2008-09-10 EP claimed
WO-2007071955-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-06-28 WO claimed
EP-1966174-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2008-09-10 EP disclosed
WO-2007071955-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-06-28 WO disclosed
EP-1761506-A1 SUBSTITUTED QUINAZOLONES AS ANTI-CANCER AGENTS AstraZeneca AB (SE) 2007-03-14 EP disclosed
WO-2005123696-A1 SUBSTITUTED QUINAZOLONES AS ANTI-CANCER AGENTS ASTRAZENECA AB (SE) 2005-12-29 WO disclosed