SCHEMBL4967912

SCHEMBL4967912

CC1CN(c2ccc(C(=O)Nc3ccc(Cl)c(Nc4ccccc4)c3)cn2)CCN1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 10/20 0.62
SMO Q99835 1/20 0.62
KCNH2 Q12809 2/20 0.45
MCHR1 Q99705 1/20 0.45
RAB9A P51151 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPK1 P28482 1/20 0.41
MAPK7 Q13164 1/20 0.41
IKBKB O14920 2/20 0.41
PIN1 Q13526 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971491 1.00 HDAC1 (0.62) HDAC1SMOKCNH2MCHR1RAB9A
SCHEMBL4971127 0.92 SMO (0.59) HDAC1SMORAB9AMAPK7IKBKB
SCHEMBL4972146 0.92 SMO (0.59) HDAC1SMORAB9AMAPK7IKBKB
SCHEMBL403080 0.92 SMO (0.70) HDAC1SMOKCNH2MCHR1RAB9A
SCHEMBL404107 0.92 SMO (0.70) HDAC1SMOKCNH2MCHR1RAB9A
SCHEMBL403079 0.92 SMO (0.70) HDAC1SMOKCNH2MCHR1RAB9A
SCHEMBL4972109 0.90 SMO (0.75) HDAC1SMOKCNH2MCHR1RAB9A
SCHEMBL4975497 0.87 KCNH2 (0.57) HDAC1SMOKCNH2RAB9ASMN1; SMN2
SCHEMBL402178 0.86 SMO (0.64) HDAC1SMORAB9ASMN1; SMN2NPC1
SCHEMBL399419 0.86 SMO (0.64) HDAC1SMORAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP claimed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO claimed
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP disclosed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO disclosed