SCHEMBL4968561

SCHEMBL4968561

O=C(NC(c1cc(F)cc(C(F)(F)F)c1)[C@@H](c1ccccc1)c1ccc(F)cc1)[C@@H](O)CC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.40
TACR1 P25103 11/20 0.38
CETP P11597 4/20 0.38
KCNH2 Q12809 3/20 0.37
ULK1 O75385 1/20 0.37
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CCR2 P41597 2/20 0.35
CCR5 P51681 1/20 0.35
ACP1 P24666 1/20 0.35
PTPN7 P35236 1/20 0.35
PTPN12 Q05209 1/20 0.35
PTPN13 Q12923 1/20 0.35
SSU72 Q9NP77 1/20 0.35
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971705 0.97 SLC6A9 (0.40) SLC6A9TACR1CETPKCNH2ULK1
SCHEMBL4968815 0.76 CETP (0.55) SLC6A9TACR1CETPKCNH2ULK1
SCHEMBL14244157 0.76 CETP (0.47) CETP
SCHEMBL4970220 0.72 CETP (0.43) SLC6A9TACR1CETPKCNH2CCR2
SCHEMBL4967551 0.72 CETP (0.43) SLC6A9TACR1CETPKCNH2CCR2
SCHEMBL4966775 0.72 CETP (0.43) SLC6A9TACR1CETPKCNH2CCR2
SCHEMBL4971054 0.72 SLC6A9 (0.36) SLC6A9TACR1CETPKCNH2ULK1
SCHEMBL757360 0.71 CETP (0.69) CETPKCNH2
SCHEMBL758409 0.71 CETP (0.69) CETPKCNH2
SCHEMBL760204 0.71 CETP (0.69) CETPKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954668-A2 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS Brystol-Myers Squibb Company (US) 2008-08-13 EP disclosed
WO-2007062308-A2 HOMO- AND HETEROCYCLIC COMPOUNDS SUITABLE AS CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed