SCHEMBL4968899

SCHEMBL4968899

Cc1nc(OC(C)CC(N)=O)nc(C)c1C(=O)N1CC2CN(c3cccc(CCC(N)=O)c3)CC2C1

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.38
HCRTR2 O43614 19/20 0.38
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698184 0.88 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL4696692 0.86 HCRTR1 (0.42) HCRTR1HCRTR2KCNH2
SCHEMBL4697094 0.83 HCRTR1 (0.40) HCRTR1HCRTR2KCNH2
SCHEMBL4809142 0.83 HCRTR1 (0.41) HCRTR1HCRTR2KCNH2
SCHEMBL4968486 0.82 HCRTR1 (0.42) HCRTR1HCRTR2KCNH2
SCHEMBL5234333 0.82 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL4696182 0.82 HCRTR1 (0.38) HCRTR1HCRTR2KCNH2
SCHEMBL4696183 0.82 HCRTR1 (0.38) HCRTR1HCRTR2KCNH2
SCHEMBL4698004 0.81 HCRTR1 (0.39) HCRTR1HCRTR2KCNH2
SCHEMBL5236658 0.80 HCRTR1 (0.40) HCRTR1HCRTR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987035-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2008-11-05 EP disclosed
WO-2007093515-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN LA-ROCHE AG (CH) 2007-08-23 WO disclosed