SCHEMBL4969703

SCHEMBL4969703

C=C(C)COc1ccc(C=O)c(F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
POLB P06746 2/20 0.42
ALDH1A1 P00352 2/20 0.42
PKM P14618 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GPR174 Q9BXC1 1/20 0.40
MAOB P27338 3/20 0.39
AOC3 Q16853 1/20 0.39
TRIM24 O15164 1/20 0.38
TYR P14679 1/20 0.38
TRIM33 Q9UPN9 1/20 0.38
ERN1 O75460 1/20 0.36
MAPK1 P28482 2/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.36
ALOX12 P18054 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464487 0.80 MAOB (0.53) MEN1KMT2APOLBALDH1A1PKM
SCHEMBL3170130 0.79 NQO1 (0.45) KMT2AALDH1A1ERN1TSHRHSD17B10
SCHEMBL11238246 0.79 KMT2A (0.45) MEN1KMT2APOLBALDH1A1PKM
SCHEMBL22322029 0.79 ALDH1A1 (0.37) POLBALDH1A1MAOBAOC3TRIM24
SCHEMBL28743714 0.78 KDM4E (0.58) POLBALDH1A1MAPK1HSD17B10MAPT
SCHEMBL3574606 0.76 PDE3B (0.43) POLBALDH1A1TRIM24TYRTRIM33
SCHEMBL8070059 0.76 MCL1 (0.42) MEN1KMT2AALDH1A1L3MBTL1ERN1
SCHEMBL1443540 0.76 ERN1 (0.47) MEN1KMT2AMAOBERN1MAPK1
SCHEMBL13862092 0.76 MAOB (0.42) MEN1KMT2APOLBALDH1A1PKM
SCHEMBL18990273 0.76 KMT2A (0.42) MEN1KMT2APOLBALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099020-A1 1,1-DIOXO-1-THIA-5,10-DIAZADIBENZOCYCLOHEPTENES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed
WO-2008099020-A1 1,1-DIOXO-1-THIA-5,10-DIAZADIBENZOCYCLOHEPTENES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed