SCHEMBL4969967

SCHEMBL4969967

CNC(C1CCCC1)C(C)NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
EPHX1 P07099 1/20 0.40
CTSK P43235 7/20 0.40
CTSS P25774 5/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
BTK Q06187 1/20 0.39
KMT2A Q03164 1/20 0.39
AAK1 Q2M2I8 1/20 0.38
CYP2D6 P10635 1/20 0.36
CTSL P07711 3/20 0.36
CTSB P07858 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971473 0.98 GAA (0.43) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL4972585 0.98 GAA (0.43) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL4971810 0.83 EPHX1 (0.43) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL9833367 0.83 CYP2D6 (0.42) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL4971674 0.83 GAA (0.44) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL22506436 0.83 GAA (0.44) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL22535888 0.83 GAA (0.44) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL20470280 0.83 GAA (0.44) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL14011490 0.81 GAA (0.47) GAAHDAC4HDAC1HDAC6EPHX1
SCHEMBL4753064 0.81 GAA (0.47) GAAHDAC4HDAC1HDAC6EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed