SCHEMBL4970569

SCHEMBL4970569

Cc1onc(-c2cccc(F)c2)c1-c1c[nH]c(-c2ccc(C(=O)NC3CCC3)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 11/20 0.51
HDAC4 P56524 2/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HPGDS O60760 1/20 0.42
GRM5 P41594 1/20 0.41
USP30 Q70CQ3 2/20 0.40
SMYD3 Q9H7B4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4971397 0.98 GABRA5 (0.51) GABRA5HDAC4HDAC6HPGDSUSP30
SCHEMBL4971020 0.97 GABRA5 (0.55) GABRA5HDAC4HPGDSUSP30SMYD3
SCHEMBL4972209 0.94 GABRA5 (0.50) GABRA5HPGDSGRM5
SCHEMBL4973770 0.92 GABRA5 (0.50) GABRA5HPGDSGRM5
SCHEMBL4971806 0.91 GABRA5 (0.53) GABRA5HPGDSGRM5
SCHEMBL4971009 0.91 GABRA5 (0.51) GABRA5HDAC4HDAC6SMYD3
SCHEMBL4971725 0.90 GABRA5 (0.49) GABRA5HDAC4HDAC6SMYD3
SCHEMBL4971711 0.89 GABRA5 (0.51) GABRA5HDAC4SMYD3
SCHEMBL4970995 0.88 GABRA5 (0.56) GABRA5
SCHEMBL4973220 0.87 MAPK14 (0.52) GABRA5SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968973-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2008-09-17 EP claimed
WO-2007074078-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-07-05 WO claimed
EP-1968973-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2008-09-17 EP disclosed
WO-2007074078-A2 ARYL-ISOXAZOL-4-YL-IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-07-05 WO disclosed