SCHEMBL4970829

SCHEMBL4970829

CCC[C@](OCCO)(c1cccc(Cl)c1)[C@@H]1CCCN(C(C)(C)C)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 11/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM2B Q8NHM5 1/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HRH3 Q9Y5N1 3/20 0.33
KDM4E B2RXH2 1/20 0.33
SLC22A1 O15245 1/20 0.33
MLNR O43193 1/20 0.33
NR1I2 O75469 1/20 0.33
TP53 P04637 1/20 0.33
ADRB2 P07550 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
ADRB1 P08588 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
CHRM5 P08912 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968765 0.86 REN (0.32) RENMEN1KMT2AKDM2BHRH3
SCHEMBL4971351 0.85 MEN1 (0.37) RENMEN1KMT2AKDM2BMAPK1
SCHEMBL8236287 0.84 REN (0.35) RENMEN1KMT2AKDM2BMAPK1
SCHEMBL3613909 0.84 REN (0.42) RENTP53
SCHEMBL3613911 0.84 REN (0.42) RENTP53
SCHEMBL4971651 0.80 MEN1 (0.35) MEN1KMT2ADRD2CHRM3SLC6A2
SCHEMBL4971952 0.77 REN (0.42) RENSCN5A
SCHEMBL27737826 0.77 REN (0.42) RENSCN5A
SCHEMBL3613379 0.76 REN (0.41) RENTP53
SCHEMBL3613375 0.76 REN (0.41) RENTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed