SCHEMBL4971105

SCHEMBL4971105

NC(=O)[C@@H]1CCCN1c1ccccc1-n1cccc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.54
ELANE P08246 2/20 0.46
MAPK1 P28482 1/20 0.46
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
OGFRL1 Q5TC84 1/20 0.42
HTR1A P08908 5/20 0.41
HTR7 P34969 5/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAT2A P31153 2/20 0.39
SCN9A Q15858 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
DPP4 P27487 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15330912 0.78 AR (0.56) ARELANEOPRM1OPRD1OPRK1
SCHEMBL15665470 0.76 ELANE (0.54) ARELANEOPRM1OPRD1OPRK1
SCHEMBL2172636 0.76 ELANE (0.54) ARELANEOPRM1OPRD1OPRK1
SCHEMBL3347621 0.76 ELANE (0.54) ARELANEOPRM1OPRD1OPRK1
SCHEMBL28510719 0.75 AR (0.50) ARELANEOPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL27002674 0.75 ELANE (0.53) ARELANEOPRM1OPRD1OPRK1
SCHEMBL5736480 0.75 ITGB3 (0.53) MAPK1ALDH1A1DPP4
SCHEMBL2555259 0.74 AR (0.52) ARELANEOPRM1OPRD1OPRK1
SCHEMBL7497512 0.72 ELANE (0.50) ARELANEOPRM1OPRD1OPRK1
SCHEMBL27534007 0.72 ELANE (0.50) ARELANEOPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888563-A1 PROLINE BIS-AMIDE OREXIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2008-02-20 EP disclosed
WO-2006127550-A1 PROLINE BIS-AMIDE OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-11-30 WO disclosed