SCHEMBL4972254

SCHEMBL4972254

O=C(Nc1ccc(Cl)c(Nc2ccccc2)c1)c1ccc(N2CCC(O)CC2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.53
MAPK8 P45983 3/20 0.46
MCHR1 Q99705 2/20 0.46
KCNH2 Q12809 2/20 0.46
DGAT1 O75907 5/20 0.45
RAB9A P51151 3/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HTT P42858 1/20 0.45
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
CYP3A4 P08684 1/20 0.43
SOAT1 P35610 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42
KCNQ3 O43525 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4969870 0.92 SMO (0.50) SMOMCHR1DGAT1RAB9ALMNA
SCHEMBL4971602 0.92 SMO (0.52) SMOMCHR1KCNH2RAB9ALMNA
SCHEMBL402625 0.91 SMO (0.60) SMOMAPK8MCHR1KCNH2DGAT1
SCHEMBL4970492 0.89 SMO (0.52) SMOMAPK8MCHR1KCNH2DGAT1
SCHEMBL4975497 0.88 KCNH2 (0.57) SMOMAPK8KCNH2RAB9ALMNA
SCHEMBL10238407 0.87 SMO (0.56) SMOALDH1A1HDAC2
SCHEMBL399857 0.87 MAPT (0.57) SMOMAPK8MCHR1RAB9ALMNA
SCHEMBL404073 0.87 SMO (0.59) SMOMAPK8MCHR1RAB9ALMNA
SCHEMBL4972268 0.86 SMO (0.52) SMORAB9ALMNAMAPTSMN1; SMN2
SCHEMBL10238332 0.85 SMO (0.58) SMORAB9ALMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957461-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING Genentech, Inc. (US) 2008-08-20 EP disclosed
WO-2007059157-A1 BISAMIDE INHIBITORS OF HEDGEHOG SIGNALING GENENTECH, INC. (US) 2007-05-24 WO disclosed