SCHEMBL4974692

SCHEMBL4974692

COc1cccc(B(O)O)c1.OB(O)c1cccc(Cl)c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 4/20 0.79
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
RELA Q04206 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
PGR P06401 2/20 0.43
NLRP3 Q96P20 1/20 0.43
EGFR P00533 1/20 0.42
ERBB3 P21860 1/20 0.42
ACHE P22303 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
NFE2L2 Q16236 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
GFER P55789 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5140 0.89 ENPP2 (1.00) ENPP2CA1CA2RELANPC1
SCHEMBL7344145 0.89 ENPP2 (1.00) ENPP2CA1CA2RELANPC1
Methyl Alcohol SCHEMBL28712606 0.87 ENPP2 (0.96) ENPP2CA1CA2RELANPC1
SCHEMBL11815 0.83 ENPP2 (0.56) ENPP2CA1CA2EGFR
SCHEMBL4974695 0.83 ENPP2 (0.54) ENPP2CA1CA2RELANPC1
SCHEMBL28060965 0.82 ENPP2 (0.85) ENPP2CA1CA2NLRP3ACHE
SCHEMBL29563391 0.82 ENPP2 (0.56) ENPP2CA1CA2LMNA
SCHEMBL29056807 0.82 ENPP2 (0.56) ENPP2CA1CA2LMNA
SCHEMBL28270052 0.81 ENPP2 (0.50) ENPP2CA1CA2RELAEGFR
Acetonitrile SCHEMBL28133848 0.81 ENPP2 (0.82) ENPP2CA1CA2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979335-A2 THIAZOLES AS 11 BETA-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2008-10-15 EP disclosed
WO-2007082808-A2 THIAZOLES AS 11 BETA-HSD1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-07-26 WO disclosed