SCHEMBL4976543

SCHEMBL4976543

CS(=O)(=O)OCC1CN(C(=O)O)CCN1Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.50
CA2 P00918 6/20 0.50
CA4 P22748 6/20 0.50
CA9 Q16790 6/20 0.50
ALDH1A1 P00352 3/20 0.43
SIGMAR1 Q99720 3/20 0.42
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.40
GAA P10253 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3493064 0.87 JAK2 (0.47) CA1CA2CA4CA9ALDH1A1
SCHEMBL24328 0.84 SIGMAR1 (0.56) ALDH1A1SIGMAR1LMNAGAA
SCHEMBL3494894 0.82 CA1 (0.48) CA1CA2CA4CA9SIGMAR1
SCHEMBL30483521 0.81 SIGMAR1 (0.40) CA1CA2CA4CA9ALDH1A1
SCHEMBL17154894 0.80 GBA1 (0.43)
SCHEMBL3495972 0.80 SIGMAR1 (0.54) CA1CA2CA4CA9ALDH1A1
SCHEMBL4971104 0.80 SIGMAR1 (0.54) CA1CA2CA4CA9ALDH1A1
SCHEMBL27533150 0.80 CA1 (0.63) CA1CA2CA4CA9
SCHEMBL20974922 0.80 SIGMAR1 (0.54) CA1CA2CA4CA9ALDH1A1
SCHEMBL26094131 0.79 CA1 (0.50) CA1CA2CA4CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed