SCHEMBL4978183

SCHEMBL4978183

COc1cc(N)nn1C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.37
NR1H2 P55055 2/20 0.35
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34
TUBB2B Q9BVA1 1/20 0.34
TUBB1 Q9H4B7 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
MAP2K4 P45985 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788542 0.84 FAAH (0.35) FAAHNR1H2HSP90AA1HSP90AB1MAP2K4
SCHEMBL25203731 0.82 FAAH (0.34) FAAHNR1H2HSP90AA1HSP90AB1MAP2K4
SCHEMBL161429 0.81 FAAH (0.39) FAAHNR1H2TUBB4ATUBBTUBA3C
SCHEMBL2480409 0.79 FAAH (0.38) FAAHNR1H2HSP90AA1HSP90AB1MAP2K4
SCHEMBL19010764 0.78 FAAH (0.38) FAAHNR1H2TUBB4ATUBBTUBA3C
SCHEMBL25519570 0.77 MAP2K4 (0.40) FAAHNR1H2HSP90AA1HSP90AB1MAP2K4
SCHEMBL18284944 0.77 FAAH (0.39) FAAHNR1H2HSP90AA1HSP90AB1MAP2K4
SCHEMBL25519814 0.77 FAAH (0.39) FAAHNR1H2HSP90AA1HSP90AB1MAP2K4
SCHEMBL2489522 0.75 ELANE (0.39) FAAHNR1H2ELANECTSDCTSE
SCHEMBL20575911 0.74 CFTR (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008132502-A1 PYRAZOLYL-AMINO-SUBSTITUTED PYRIMIDINES AND THEIR USE FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-11-06 WO disclosed