SCHEMBL4979414

SCHEMBL4979414

CC1(C)Oc2cc(NS(C)(=O)=O)[c]cc2N(c2ccc(F)cc2)C1=O

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 6/20 0.71
BRD4 O60885 4/20 0.38
AR P10275 1/20 0.34
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34
SCN9A Q15858 1/20 0.33
TP53 P04637 1/20 0.32
PGR P06401 1/20 0.32
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mt-3995 SCHEMBL753911 0.83 NR3C2 (1.00) NR3C2BRD4ARPTGS2
SCHEMBL754239 0.80 NR3C2 (0.71) NR3C2BRD4ARCACNA1BAPBA1
SCHEMBL755189 0.80 NR3C2 (0.70) NR3C2BRD4ARCACNA1BAPBA1
SCHEMBL755350 0.80 NR3C2 (0.70) NR3C2BRD4ARCACNA1BAPBA1
SCHEMBL761147 0.80 NR3C2 (0.70) NR3C2BRD4ARCACNA1BAPBA1
SCHEMBL2266367 0.78 NR3C2 (0.67) NR3C2BRD4SCN9APGR
SCHEMBL2269447 0.77 NR3C2 (0.69) NR3C2ARCACNA1BAPBA1LMNA
SCHEMBL755391 0.77 NR3C2 (0.72) NR3C2BRD4ARCACNA1BAPBA1
SCHEMBL4530965 0.76 NR3C2 (0.65) NR3C2BRD4SCN9A
SCHEMBL755900 0.76 NR3C2 (0.71) NR3C2BRD4ARCACNA1BAPBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984345-A1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS Mitsubishi Tanabe Pharma Corporation (JP) 2008-10-29 EP disclosed
WO-2007089034-A1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-08-09 WO disclosed