SCHEMBL4979423

SCHEMBL4979423

CN1CCN(c2ccc(-c3ccccc3CCN(c3cccnc3)c3cccnc3)cn2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CLK4 Q9HAZ1 1/20 0.41
ACVR1B P36896 1/20 0.41
TGFBR1 P36897 1/20 0.41
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
FYN P06241 2/20 0.39
TDO2 P48775 1/20 0.39
TNKS O95271 1/20 0.38
ATR Q13535 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
CNR2 P34972 1/20 0.37
EED O75530 1/20 0.37
SUZ12 Q15022 1/20 0.37
EZH2 Q15910 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4974371 0.78 KCNA5 (0.50) CYP3A4ALDH1A1CYP1A2TSHRHSD17B10
SCHEMBL884336 0.78 KCNA5 (0.60) CYP3A4ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL1368757 0.77 ALDH1A1 (0.42) CYP3A4ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL4975470 0.74 KCNA5 (0.51) ALDH1A1TSHR
SCHEMBL10094621 0.70 CYP1A2 (0.57) CYP3A4ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL3241755 0.69 CNR2 (0.56) ALDH1A1ACVR1BTGFBR1BRD4CREBBP
SCHEMBL3623417 0.69 PDK2 (0.42) ALDH1A1
SCHEMBL15784005 0.67 ATR (0.52) CYP3A4ALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL10094346 0.67 FYN (0.48) ACVR1BTGFBR1BRD4CREBBPFYN
SCHEMBL884799 0.67 KCNA5 (0.52) CYP3A4ALDH1A1CYP1A2CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed