SCHEMBL4980452

SCHEMBL4980452

Cc1c[nH]c(=O)c2ccc(OC3CCCN(C(=O)O)C3)cc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.61
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
SPR P35270 1/20 0.41
PARP1 P09874 4/20 0.39
HRH1 P35367 1/20 0.39
CCR3 P51677 1/20 0.39
CYP4A11 Q02928 2/20 0.39
CYP4F2 P78329 1/20 0.39
ROCK2 O75116 1/20 0.38
PRKX P51817 1/20 0.38
PRKCE Q02156 1/20 0.38
PRKCD Q05655 1/20 0.38
PRKD1 Q15139 1/20 0.38
CHEK2 O96017 1/20 0.37
HTR6 P50406 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4980445 1.00 ROCK1 (0.61) ROCK1MTNR1AMTNR1BHCRTR1HCRTR2
SCHEMBL4968833 0.88 ROCK1 (0.45) ROCK1MTNR1AMTNR1BHCRTR1HCRTR2
SCHEMBL4968824 0.88 ROCK1 (0.45) ROCK1MTNR1AMTNR1BHCRTR1HCRTR2
SCHEMBL4007663 0.87 ROCK1 (0.56) ROCK1MTNR1AMTNR1BHCRTR1HCRTR2
SCHEMBL4007667 0.87 ROCK1 (0.56) ROCK1MTNR1AMTNR1BHCRTR1HCRTR2
SCHEMBL4965892 0.81 ROCK1 (0.59) ROCK1ROCK2PRKXPRKCEPRKCD
SCHEMBL4965898 0.81 ROCK1 (0.59) ROCK1ROCK2PRKXPRKCEPRKCD
SCHEMBL8938507 0.81 ROCK1 (0.76) ROCK1PARP1ROCK2PRKXPRKCE
SCHEMBL30283494 0.79 MTNR1A (0.46) ROCK1MTNR1AMTNR1BHCRTR1HCRTR2
SCHEMBL4009155 0.77 CHEK2 (0.48) ROCK1MTNR1AMTNR1BCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963304-A1 ISOQUINOLINE DERIVATIVES N.V. Organon (NL) 2008-09-03 EP disclosed
WO-2007065916-A1 ISOQUINOLINE DERIVATIVES N.V. ORGANON (NL) 2007-06-14 WO disclosed