SCHEMBL4982251

SCHEMBL4982251

CC(C)(C)C(c1ccccc1)[C@@H]1CN(C(=O)O)CCN1C(=O)c1ncn(-c2cccc(OCc3ccccc3)c2)c1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.38
MGLL Q99685 3/20 0.36
ALDH1A1 P00352 2/20 0.35
CCKAR P32238 1/20 0.35
SPHK2 Q9NRA0 2/20 0.34
SPHK1 Q9NYA1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
BTK Q06187 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTSA P10619 1/20 0.33
CHRM3 P20309 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3494934 0.88 POLB (0.36) MGLLALDH1A1SPHK2LMNAKMT2A
SCHEMBL3494754 0.88 POLB (0.36) MGLLALDH1A1SPHK2LMNAKMT2A
SCHEMBL3492728 0.83 SPHK2 (0.41) FAAHMGLLALDH1A1SPHK2SPHK1
SCHEMBL3493899 0.82 DHODH (0.36) MGLLALDH1A1SPHK2SPHK1KDM4E
SCHEMBL3494080 0.81 MDM2 (0.38) KDM4EMAPT
SCHEMBL4982247 0.79 ABHD6 (0.46) FAAHMGLLSPHK2
SCHEMBL3492193 0.77 AVPR2 (0.39) MGLLALDH1A1KMT2A
SCHEMBL3491863 0.74 CA1 (0.40)
SCHEMBL3495945 0.72 NOTUM (0.34) FAAHALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL4978695 0.72 CYP2D6 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed