SCHEMBL4982702

SCHEMBL4982702

Cc1cccc(C(=O)N=S=O)c1-c1ncc[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.44
TYRO3 Q06418 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
PARP1 P09874 1/20 0.39
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 3/20 0.38
KMT2A Q03164 2/20 0.35
NISCH Q9Y2I1 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
MYC P01106 1/20 0.33
MTOR P42345 1/20 0.33
ADK P55263 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4564863 0.81 CSNK1A1 (0.61) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
SCHEMBL29054844 0.81 CSNK1A1 (0.50) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
SCHEMBL6001368 0.75 NISCH (0.52) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
Hydrochloric Acid SCHEMBL29265356 0.74 NISCH (0.50) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
SCHEMBL28766417 0.71 NISCH (0.47) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
SCHEMBL14886293 0.71 CSNK1A1 (0.54) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
SCHEMBL11813949 0.70 HPGD (0.43) ALDH1A1KDM4EKMT2AMYCHPGD
SCHEMBL9260794 0.70 NISCH (0.46) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1
SCHEMBL19782078 0.68 NISCH (0.44) CSNK1A1TYRO3DYRK1BALDH1A1KDM4E
SCHEMBL28348460 0.66 CSNK1A1 (0.60) CSNK1A1TYRO3DYRK1BPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976835-A2 HISTONE DEACETYLASE INHIBITORS Takeda San Diego, Inc. (US) 2008-10-08 EP disclosed
WO-2007084390-A2 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2007-07-26 WO disclosed