SCHEMBL499157

SCHEMBL499157

CN[C@H](CNC(=O)N(C)CC[C@@H](OCCN(C)C(=O)O)c1cccc(Cl)c1)C[C@H]1CCCCOC1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 17/20 0.52
CYP3A4 P08684 3/20 0.46
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499595 0.98 REN (0.54) RENCYP3A4ALDH1A1GAAL3MBTL1
SCHEMBL4789610 0.92 REN (0.55) RENCYP3A4ALDH1A1GAAL3MBTL1
SCHEMBL499779 0.92 REN (0.55) RENCYP3A4ALDH1A1GAAL3MBTL1
SCHEMBL499038 0.91 REN (0.47) RENCYP3A4ALDH1A1GAAL3MBTL1
SCHEMBL10254125 0.90 REN (0.63) RENCYP3A4
SCHEMBL499005 0.90 REN (0.52) RENCYP3A4
SCHEMBL3334092 0.90 REN (0.57) RENCYP3A4ALDH1A1GAAL3MBTL1
SCHEMBL497543 0.90 REN (0.52) RENCYP3A4
SCHEMBL10253693 0.88 REN (0.65) RENCYP3A4
SCHEMBL499022 0.88 REN (0.54) RENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US claimed
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed