⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL7072086 | 0.86 | — | — | |
| SCHEMBL10542818 | 0.78 | KDM4E (0.33) | — | |
| Hydrochloric Acid SCHEMBL3237965 | 0.77 | — | — | |
| SCHEMBL4721663 | 0.75 | — | — | |
| SCHEMBL1193464 | 0.75 | — | — | |
| SCHEMBL5204363 | 0.70 | — | — | |
| SCHEMBL15047584 | 0.70 | — | — | |
| SCHEMBL9244035 | 0.70 | — | — | |
| SCHEMBL19599281 | 0.67 | — | — | |
| SCHEMBL3816759 | 0.67 | AGL (0.30) | — |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-0304552-A1 | Heterocyclic hydroxyazoles | BAYER AG (DE) | 1989-03-01 | — | — | EP | claimed |
| EP-0011769-B1 | HYDROXYETHYL AZOLES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MEDICAMENTS | BAYER AG (DE) | 1982-04-14 | — | — | EP | claimed |
| EP-0017080-A2 | Process for the preparation of hydroxyethyl azoles; intermediates | BAYER AG (DE) | 1980-10-15 | — | — | EP | claimed |
| EP-0011769-A1 | Hydroxyethyl azoles, process for their preparation and their use in medicaments | BAYER AG (DE) | 1980-06-11 | — | — | EP | claimed |
| CN-119548497-A | Method for treating myopia by using vinpocetine | 温州医科大学附属眼视光医院 | 2025-03-04 | — | — | CN | disclosed |
| CN-119061713-A | Recording method and composition set | 精工爱普生株式会社 | 2024-12-03 | — | — | CN | disclosed |
| CN-118634218-A | Pharmaceutical composition for effectively delaying and treating myopia | 温州医科大学附属眼视光医院 | 2024-09-13 | — | — | CN | disclosed |
| US-20240165089-A1 | METHOD FOR TREATING MYOPIA WITH VINPOCETINE | Eye Hospital, Wenzhou Medical University (CN) | 2024-05-23 | — | — | US | disclosed |
| EP-4364736-A1 | METHOD FOR TREATING MYOPIA WITH VINPOCETINE | The Eye Hospital of Wenzhou Medical University (CN) | 2024-05-08 | — | — | EP | disclosed |
| CN-113015526-A | Spirocyclic 2, 3-dihydro-7-azaindole compounds and uses thereof | 豪夫迈·罗氏有限公司 | 2021-06-22 | — | — | CN | disclosed |
| US-20150112051-A1 | CONSTRUCTION OF CELL PENETRATING NUCLEIC ACIDS | Panzner, Steffen | 2015-04-23 | — | — | US | disclosed |
| US-20150112051-A1 | CONSTRUCTION OF CELL PENETRATING NUCLEIC ACIDS | Panzner, Steffen | 2015-04-23 | — | — | US | disclosed |
| US-20030199478-A1 | 3-(Arylamino)methylene-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors | ALLERGAN, INC. | 2003-10-23 | — | — | US | disclosed |
| WO-2003027102-A1 | 3-(ARYLAMINO)METHYLENE-1, 3-DIHYDRO-2H-INDOL-2-ONES AS KINASE INHIBITORS | ALLERGAN, INC. (US) | 2003-04-03 | — | — | WO | disclosed |
| EP-0304552-A1 | Heterocyclic hydroxyazoles | BAYER AG (DE) | 1989-03-01 | — | — | EP | disclosed |
| EP-0304552-A1 | Heterocyclic hydroxyazoles | BAYER AG (DE) | 1989-03-01 | — | — | EP | disclosed |
| EP-0017080-A3 | PROCESS FOR THE PREPARATION OF HYDROXYETHYL AZOLES; INTERMEDIATES | BAYER AG (DE) | 1981-01-14 | — | — | EP | disclosed |
| EP-0017080-A2 | Process for the preparation of hydroxyethyl azoles; intermediates | BAYER AG (DE) | 1980-10-15 | — | — | EP | disclosed |
| EP-0017080-A2 | Process for the preparation of hydroxyethyl azoles; intermediates | BAYER AG (DE) | 1980-10-15 | — | — | EP | disclosed |
| EP-0011769-A1 | Hydroxyethyl azoles, process for their preparation and their use in medicaments | BAYER AG (DE) | 1980-06-11 | — | — | EP | disclosed |