SCHEMBL4992908

SCHEMBL4992908

Nc1nc(NCCNc2ncc(-c3cnc[nH]3)c(-c3ccccc3)n2)ccc1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.53
GSK3A P49840 3/20 0.53
CDK1 P06493 2/20 0.53
CCNB2 O95067 1/20 0.53
CCNB1 P14635 1/20 0.53
CCNB3 Q8WWL7 1/20 0.53
ADORA1 P30542 3/20 0.38
MAPT P10636 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PRKCQ Q04759 2/20 0.34
DHFR P00374 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4395953 0.90 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4393950 0.89 GSK3B (0.50) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4992921 0.84 GSK3B (0.73) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4394516 0.84 GSK3B (0.76) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL7658642 0.78 GSK3B (0.46) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL7024960 0.78 ADORA1 (0.48) ADORA1HPGD
SCHEMBL7256594 0.76 GSK3B (0.50) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL5100038 0.76 GSK3B (0.82) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL5100682 0.75 GSK3B (0.64) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL7255038 0.75 GSK3B (0.49) GSK3BMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1653970-A4 GSK-3 INHIBITORS AND USES THEREOF NOVARTIS VACCINES & DIAGNOSTIC (US) 2008-10-15 EP disclosed
EP-1653970-A2 GSK-3 INHIBITORS AND USES THEREOF CHIRON CORPORATION (US) 2006-05-10 EP disclosed
WO-2005039485-A2 GSK-3 INHIBITORS AND USES THEREOF CHIRON CORPORATION (US) 2005-05-06 WO disclosed