SCHEMBL7024960

SCHEMBL7024960

NCCNc1ncc(-c2cnc[nH]2)c(-c2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.48
IDO1 P14902 8/20 0.43
CYP3A4 P08684 1/20 0.43
SYK P43405 2/20 0.41
ZAP70 P43403 1/20 0.41
HPGDS O60760 1/20 0.41
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
NAMPT P43490 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024964 0.79 ADORA1 (0.46) ADORA1SYKZAP70KDM4EALDH1A1
SCHEMBL4992908 0.78 GSK3B (0.53) ADORA1HPGD
SCHEMBL5099790 0.73 KDM1A (0.40) ADORA1IDO1
SCHEMBL5100481 0.72 GSK3B (0.48) IDO1CYP3A4
SCHEMBL27722304 0.69 ADORA1 (0.52) ADORA1
SCHEMBL7211775 0.68 PTGS2 (0.48) ADORA1ADORA2A
SCHEMBL5089828 0.68 GSK3B (0.44) ADORA1IDO1CYP3A4
SCHEMBL7256594 0.68 GSK3B (0.50) ALDH1A1GAAMKNK1
Hydrochloric Acid SCHEMBL7210504 0.68 PTGS2 (0.47) ADORA1ADORA2A
SCHEMBL5094245 0.67 CCNB2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed