SCHEMBL5003263

SCHEMBL5003263

COc1cc(-c2ccc(C(=O)C(C)C(C)(C)C(=O)O)cc2)ccc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.48
ABCB1 P08183 8/20 0.44
ABCC1 P33527 5/20 0.43
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5007308 0.81 ALDH1A1 (0.51) CHEK1ABCB1ABCC1ALDH1A1CYP3A4
SCHEMBL6030795 0.80 CHEK1 (0.48) CHEK1ABCB1ABCC1CYP3A4
SCHEMBL4525042 0.80 CHEK1 (0.46) CHEK1ABCB1ABCC1
SCHEMBL11224598 0.76 CHEK1 (0.61) CHEK1ABCB1ABCC1ALDH1A1CYP3A4
SCHEMBL30423771 0.75 ALDH1A1 (0.61) CHEK1ABCB1ABCC1ALDH1A1TDP1
SCHEMBL359057 0.75 ALDH1A1 (0.61) CHEK1ABCB1ABCC1ALDH1A1TDP1
SCHEMBL1747968 0.74 NPC1 (0.45) CHEK1ABCB1ABCC1CYP3A4
SCHEMBL16701438 0.74 CHEK1 (0.54) CHEK1ABCB1ABCC1ALDH1A1TDP1
SCHEMBL223878 0.72 TTR (0.64) ALDH1A1TSHR
SCHEMBL29753668 0.72 TTR (0.64) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423156-B2 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER PHARMACEUTICALS CORPORATION (US) 2008-09-09 US disclosed