SCHEMBL5009745

SCHEMBL5009745

NC(=O)C1(c2ccc(-c3ccc(CC(N)(F)F)cc3)c(F)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 10/20 0.55
CYP2C9 P11712 7/20 0.51
CYP2C19 P33261 6/20 0.51
CYP3A4 P08684 6/20 0.51
CYP2D6 P10635 3/20 0.51
AKR1C3 P42330 6/20 0.49
AKR1C2 P52895 6/20 0.49
AKR1C1 Q04828 3/20 0.49
CTSK P43235 2/20 0.47
AKR1B10 O60218 1/20 0.46
AKR1C4 P17516 1/20 0.46
PSEN1 P49768 1/20 0.46
PSEN2 P49810 1/20 0.46
APH1B Q8WW43 1/20 0.46
NCSTN Q92542 1/20 0.46
APH1A Q96BI3 1/20 0.46
PSENEN Q9NZ42 1/20 0.46
CYP1A2 P05177 1/20 0.43
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011741 0.91 APP (0.55) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL5014679 0.85 SYK (0.42) APPCYP2C9CYP2C19CYP2D6CTSK
SCHEMBL4505580 0.79 APP (0.55) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4513813 0.79 APP (0.55) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4498009 0.78 APP (0.60) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL5181860 0.75 APP (0.55) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4514275 0.75 APP (0.52) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL4513629 0.75 APP (0.52) APPCYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL5009692 0.74 APP (0.56) APPCYP2C9CYP3A4AKR1C3AKR1C2
SCHEMBL5011694 0.74 SYK (0.42) APPCYP2C9CYP2C19CYP2D6CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed