SCHEMBL5009692

SCHEMBL5009692

CC(C)(C(N)=O)c1ccc(-c2ccc(CC(N)(F)F)cc2)c(F)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.56
AKR1C3 P42330 4/20 0.46
AKR1C2 P52895 4/20 0.46
RORC P51449 12/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011613 0.90 APP (0.56) APPAKR1C3AKR1C2RORCCYP3A4
SCHEMBL4494820 0.77 APP (0.56) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL4498505 0.75 APP (0.54) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL4501897 0.74 APP (0.53) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL5009745 0.74 APP (0.55) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL5011544 0.69 RORC (0.46) APPRORCPSEN1PSEN2APH1B
SCHEMBL8755138 0.69 APP (0.78) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL3938352 0.69 APP (0.78) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL29130916 0.68 MAPT (0.47) APPAKR1C3AKR1C2CYP3A4CYP2C9
SCHEMBL24031016 0.67 RORC (0.51) APPAKR1C3AKR1C2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed