SCHEMBL5010553

SCHEMBL5010553

O=c1cc(-c2ccc(F)cc2)c2ccc(Sc3ncc(C(O)(c4ccc(Cl)cc4)C(F)(F)F)s3)cc2o1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 7/20 0.59
MLYCD O95822 2/20 0.55
CA12 O43570 6/20 0.42
CA9 Q16790 6/20 0.42
MAPK14 Q16539 1/20 0.32
ALDH2 P05091 1/20 0.31
AKR1B1 P15121 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
HSD17B3 P37058 1/20 0.31
SORD Q00796 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2979741 0.97 MLYCD (0.58) ALOX5MLYCDCA12CA9ALDH2
SCHEMBL2983368 0.93 MLYCD (0.56) ALOX5MLYCDCA12CA9ALDH2
SCHEMBL2991946 0.87 MLYCD (0.71) ALOX5MLYCDCA12CA9ALDH2
SCHEMBL2990446 0.85 MLYCD (0.59) ALOX5MLYCDCA12CA9ALDH2
SCHEMBL2987971 0.85 MLYCD (0.65) ALOX5MLYCDCA12CA9
SCHEMBL2979837 0.83 MLYCD (0.57) ALOX5MLYCDCA12CA9
SCHEMBL2984933 0.83 MLYCD (0.57) ALOX5MLYCDCA12CA9
SCHEMBL2985044 0.83 MLYCD (0.57) ALOX5MLYCDCA12CA9
SCHEMBL2982483 0.83 MLYCD (0.57) ALOX5MLYCDCA12CA9
SCHEMBL2987497 0.83 MLYCD (0.57) ALOX5MLYCDCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439260-B2 7-(1,3-thiazol-2-YL)thio-coumarin derivatives and their use as leukotriene biosynthesis inhibitors MERCK FORSST CANADA & CO. (CA) 2008-10-21 US disclosed
EP-1636222-A1 7-[(1,3-THIAZOL-2-YL)THIO]-COUMARIN DERIVATIVES AND THEIR USE AS LEUKOTRIENE BIOSYNTHESIS INHIBITORS Merck Frosst Canada Ltd. (CA) 2006-03-22 EP disclosed
WO-2004108720-A1 7- (1, 3-THIAZOL-2-YL)THIO!-COUMARIN DERIVATIVES AND THEIR USE AS LEUKOTRIENE BIOSYNTHESIS INHIBITORS MERCK FROSST CANADA LTD. (CA) 2004-12-16 WO disclosed