SCHEMBL5011353

SCHEMBL5011353

CC(N)Cc1ccc(-c2ccc(C3(C#N)CC3)cc2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 3/20 0.41
DPP4 P27487 2/20 0.38
CTSK P43235 2/20 0.36
CYP3A4 P08684 4/20 0.35
HSD11B1 P28845 2/20 0.35
APP P05067 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP1A2 P05177 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011393 0.88 PRKCE (0.43) FFAR4DPP4CTSKCYP3A4HSD11B1
SCHEMBL4508572 0.84 FFAR4 (0.42) FFAR4CTSKCYP3A4APPCYP2C19
SCHEMBL4491283 0.82 FFAR4 (0.45) FFAR4CYP3A4APPCYP2C19CYP2C9
SCHEMBL4514618 0.81 CYP3A4 (0.40) CTSKCYP3A4HSD11B1APPCYP2C19
SCHEMBL4514062 0.80 FFAR4 (0.48) FFAR4CYP3A4APPCYP2C19CYP2C9
SCHEMBL4503949 0.79 OPRM1 (0.47) FFAR4CYP3A4APPCYP2C19CYP2C9
SCHEMBL4512900 0.79 CYP2C19 (0.40) FFAR4CTSKCYP3A4HSD11B1APP
SCHEMBL4497508 0.79 FFAR4 (0.41) FFAR4CTSKCYP3A4HSD11B1APP
SCHEMBL5013478 0.77 APP (0.42) FFAR4CTSKCYP3A4APPCYP2C19
SCHEMBL4506497 0.77 FFAR4 (0.44) FFAR4CTSKCYP3A4HSD11B1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed