SCHEMBL5014677

SCHEMBL5014677

O=C(Nc1ccc(-c2ccc(C(O)C(F)(F)F)nc2)c(F)c1)C1CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 12/20 0.52
DHODH Q02127 2/20 0.46
PARP1 P09874 1/20 0.45
MAPT P10636 3/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
F10 P00742 1/20 0.43
GSK3B P49841 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011615 0.87 ABL1 (0.52) ABL1MAPTNPC1RAB9AGSK3B
SCHEMBL5011739 0.74 DHODH (0.49) ABL1DHODHPARP1MAPTNPC1
SCHEMBL5011321 0.73 ABL1 (0.48) ABL1DHODHPARP1MAPTNPC1
SCHEMBL5009744 0.71 DHODH (0.50) ABL1DHODHPARP1MAPTNPC1
SCHEMBL4500620 0.71 APP (0.48)
SCHEMBL17236518 0.71 DHODH (0.52) ABL1DHODHPARP1MAPTNPC1
SCHEMBL14244797 0.68 ABL1 (1.00) ABL1
SCHEMBL14244796 0.68 ABL1 (1.00) ABL1
SCHEMBL14245297 0.68 ABL1 (1.00) ABL1
SCHEMBL26633318 0.67 JAK2 (0.40) ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed