SCHEMBL5009744

SCHEMBL5009744

NC(c1ccc(-c2ccc(NC(=O)C3CC3)cc2F)cc1)C(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.50
PARP1 P09874 2/20 0.50
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
F10 P00742 2/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
NPSR1 Q6W5P4 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
PTPN1 P18031 1/20 0.41
ABL1 P00519 1/20 0.40
BACE1 P56817 1/20 0.40
MAPK14 Q16539 1/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011739 0.87 DHODH (0.49) DHODHPARP1MAPTSMN1; SMN2ALDH1A1
SCHEMBL5014676 0.85 PTPN1 (0.56) MAPTSMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL5011321 0.76 ABL1 (0.48) DHODHPARP1MAPTSMN1; SMN2ALDH1A1
SCHEMBL17236518 0.74 DHODH (0.52) DHODHPARP1MAPTSMN1; SMN2ALDH1A1
SCHEMBL5014677 0.71 ABL1 (0.52) DHODHPARP1MAPTSMN1; SMN2ALDH1A1
SCHEMBL5011692 0.71 PTPN1 (0.58) MAPTSMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL5011675 0.70 PTPN1 (0.47) MAPTKMT2AMEN1NPSR1HDAC1
SCHEMBL4498505 0.69 APP (0.54) MAPTKMT2AMEN1HPGDLMNA
SCHEMBL4514275 0.69 APP (0.52)
SCHEMBL12558144 0.69 NPC1 (0.58) MAPTSMN1; SMN2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP claimed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO claimed
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed