SCHEMBL5019486

SCHEMBL5019486

Bc1c[nH]c2ncnc(Cl)c12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.61
NOTUM Q6P988 1/20 0.40
AURKA O14965 2/20 0.36
AKT1 P31749 5/20 0.35
STK3 Q13188 6/20 0.33
STK4 Q13043 3/20 0.33
DYRK1A Q13627 3/20 0.33
TRPA1 O75762 1/20 0.33
LRRK2 Q5S007 6/20 0.33
MAP3K7 O43318 2/20 0.33
TAB1 Q15750 2/20 0.33
ROCK2 O75116 3/20 0.32
PRKD3 O94806 3/20 0.32
MAP4K4 O95819 3/20 0.32
CDK1 P06493 3/20 0.32
PHKG2 P15735 3/20 0.32
PRKACA P17612 3/20 0.32
RPS6KB1 P23443 3/20 0.32
CDK2 P24941 3/20 0.32
MARK3 P27448 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2321413 0.80 CHEK1 (0.61) CHEK1NOTUMAURKAAKT1STK3
SCHEMBL1598149 0.79 CHEK1 (0.66) CHEK1NOTUMAURKAAKT1TRPA1
SCHEMBL31329069 0.79 CHEK1 (0.66) CHEK1NOTUMAURKAAKT1TRPA1
SCHEMBL153752 0.78 CHEK1 (0.63) CHEK1NOTUMAURKAAKT1STK3
SCHEMBL2323682 0.78 CHEK1 (0.63) CHEK1NOTUMAURKAAKT1STK3
SCHEMBL154600 0.76 CHEK1 (0.61) CHEK1NOTUMAURKAAKT1DYRK1A
SCHEMBL61206 0.76 CHEK1 (1.00) CHEK1NOTUMAURKAAKT1STK3
SCHEMBL357993 0.76 CHEK1 (0.61) CHEK1NOTUMAURKAAKT1TRPA1
SCHEMBL3236479 0.76 CHEK1 (0.56) CHEK1NOTUMAURKASTK3STK4
SCHEMBL155227 0.74 CHEK1 (0.54) CHEK1NOTUMMAP3K7TAB1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013012915-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC. (US) 2013-01-24 WO disclosed
WO-2012064973-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed
WO-2011146882-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INTELLIKINE, INC. (US) 2011-11-24 WO disclosed