SCHEMBL5020125

SCHEMBL5020125

CCOC(=O)[C@H](CS)NC(=O)[C@H](Cc1ccccc1)NC(=O)CC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 2/20 0.55
TP53 P04637 1/20 0.50
MMP8 P22894 1/20 0.49
MME P08473 5/20 0.46
TACR1 P25103 1/20 0.46
ALDH1A1 P00352 1/20 0.46
THRB P10828 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
NOD2 Q9HC29 1/20 0.46
ACE P12821 1/20 0.45
CPA1 P15085 1/20 0.45
ACE2 Q9BYF1 1/20 0.45
CTSL P07711 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9487298 0.87 TP53 (0.61) PSMB5TP53MMP8TACR1ALDH1A1
SCHEMBL9487303 0.87 TP53 (0.61) PSMB5TP53MMP8TACR1ALDH1A1
SCHEMBL30481165 0.86 MME (0.58) PSMB5MMEACECPA1ACE2
SCHEMBL7617954 0.83 PSMB5 (0.50) PSMB5TP53MMP8TACR1ALDH1A1
SCHEMBL3701701 0.83 PSMB5 (0.50) PSMB5TP53MMP8TACR1ALDH1A1
SCHEMBL8848739 0.82 MMP8 (0.51) MMP8MME
SCHEMBL17619379 0.82 CNR2 (0.52) TP53ALDH1A1CTSLCTSBCTSS
SCHEMBL7923964 0.82 TP53 (0.59) TP53MMP8TACR1ALDH1A1
SCHEMBL15692319 0.82 PSMB5 (0.64) PSMB5MMEHDAC3HDAC4HDAC1
SCHEMBL7615217 0.81 PSMB5 (0.48) PSMB5TP53HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065102-A2 S-T-BUTYL PROTECTED CYSTEINE DI-PEPTIDE ANALOGS AND RELATED COMPOUNDS PROMENTIS PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed