SCHEMBL5020932

SCHEMBL5020932

CNc1nc(Nc2cn(C3CCOCC3)nc2C)ncc1N

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 18/20 0.59
CYP1A2 P05177 3/20 0.45
MAP3K14 Q99558 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5021248 0.89 LRRK2 (0.56) LRRK2MAP3K14JAK2JAK1TYK2
SCHEMBL9930430 0.85 LRRK2 (0.56) LRRK2CYP1A2MAP3K14
SCHEMBL5021351 0.85 LRRK2 (0.75) LRRK2CYP1A2
SCHEMBL19433960 0.82 LRRK2 (0.61) LRRK2CYP1A2
SCHEMBL19433957 0.81 LRRK2 (0.65) LRRK2CYP1A2
SCHEMBL5021209 0.81 LRRK2 (0.51) LRRK2CYP1A2
SCHEMBL10286423 0.81 LRRK2 (0.72) LRRK2CYP1A2MAP3K14
SCHEMBL4558665 0.79 LRRK2 (0.78) LRRK2CYP1A2
SCHEMBL28442602 0.78 LRRK2 (0.61) LRRK2MAP3K14
SCHEMBL5021249 0.78 LRRK2 (0.48) LRRK2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed