SCHEMBL5020948

SCHEMBL5020948

CNc1nc(Nc2cn(C(C)(C)N)nc2C)ncc1Cl

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 20/20 0.54
CYP1A2 P05177 4/20 0.54
TTK P33981 1/20 0.54
JAK2 O60674 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21613978 0.90 LRRK2 (0.56) LRRK2CYP1A2TTKJAK2
SCHEMBL4536356 0.86 LRRK2 (0.73) LRRK2CYP1A2TTK
SCHEMBL5021149 0.82 LRRK2 (0.54) LRRK2CYP1A2TTK
SCHEMBL4561095 0.81 LRRK2 (0.67) LRRK2CYP1A2JAK2
SCHEMBL9930742 0.78 LRRK2 (0.56) LRRK2CYP1A2TTK
SCHEMBL4561033 0.78 LRRK2 (0.69) LRRK2CYP1A2JAK2
SCHEMBL4561628 0.78 LRRK2 (0.69) LRRK2CYP1A2JAK2
SCHEMBL4561111 0.76 LRRK2 (0.55) LRRK2CYP1A2JAK2
SCHEMBL18455080 0.76 LRRK2 (0.52) LRRK2CYP1A2TTKJAK2
SCHEMBL18455174 0.74 LRRK2 (0.80) LRRK2CYP1A2TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed