SCHEMBL5021149

SCHEMBL5021149

COc1nc(Nc2cn(C(C)(C)N)nc2C)ncc1Cl

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 20/20 0.54
CYP1A2 P05177 1/20 0.41
TTK P33981 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18426442 0.91 LRRK2 (0.56) LRRK2CYP1A2TTK
SCHEMBL4540735 0.85 LRRK2 (0.52) LRRK2
SCHEMBL4536584 0.85 LRRK2 (0.72) LRRK2CYP1A2TTK
SCHEMBL5020948 0.82 LRRK2 (0.54) LRRK2CYP1A2TTK
SCHEMBL4532653 0.82 LRRK2 (0.50) LRRK2CYP1A2
SCHEMBL27939020 0.81 LRRK2 (0.50) LRRK2
SCHEMBL5021158 0.79 LRRK2 (0.55) LRRK2CYP1A2
SCHEMBL4537107 0.79 LRRK2 (0.58) LRRK2CYP1A2
SCHEMBL4539554 0.79 LRRK2 (0.53) LRRK2CYP1A2
SCHEMBL5021150 0.78 LRRK2 (0.46) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed