SCHEMBL5021023

SCHEMBL5021023

CNc1nc(Nc2cnn(C3CCOCC3)c2Cl)ncc1N

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 19/20 0.62
KCNH2 Q12809 2/20 0.45
CYP1A2 P05177 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10286423 0.88 LRRK2 (0.72) LRRK2KCNH2CYP1A2
SCHEMBL9284774 0.84 LRRK2 (0.82) LRRK2CYP1A2
SCHEMBL5020951 0.84 LRRK2 (0.80) LRRK2CYP1A2
SCHEMBL5021174 0.78 LRRK2 (0.58) LRRK2KCNH2
SCHEMBL5020932 0.77 LRRK2 (0.59) LRRK2CYP1A2
SCHEMBL16469033 0.76 LRRK2 (1.00) LRRK2
SCHEMBL4564821 0.76 LRRK2 (0.73) LRRK2CYP1A2
SCHEMBL4561209 0.73 LRRK2 (0.79) LRRK2CYP1A2
SCHEMBL5021011 0.73 LRRK2 (0.56) LRRK2KCNH2CYP1A2
SCHEMBL25951749 0.73 LRRK2 (0.70) LRRK2KCNH2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed