SCHEMBL5021172

SCHEMBL5021172

COc1nc(Nc2cnn(-c3ccc(N)cc3)c2C)ncc1Cl

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.48
LRRK2 Q5S007 12/20 0.48
ALK Q9UM73 2/20 0.39
INSR P06213 1/20 0.39
FLT3 P36888 2/20 0.39
NPBWR1 P48145 1/20 0.36
MCHR1 Q99705 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4538610 0.89 LRRK2 (0.47) EGFRLRRK2ALKINSR
SCHEMBL18454684 0.87 LRRK2 (0.44) EGFRLRRK2ALKINSR
SCHEMBL4539233 0.86 LRRK2 (0.48) EGFRLRRK2ALKINSR
SCHEMBL5021360 0.85 LRRK2 (0.64) EGFRLRRK2ALK
SCHEMBL21613957 0.85 LRRK2 (0.45) EGFRLRRK2ALKINSR
SCHEMBL4542755 0.83 LRRK2 (0.52) LRRK2
SCHEMBL5021367 0.79 EGFR (0.48) EGFRLRRK2ALKINSRFLT3
SCHEMBL4537127 0.78 LRRK2 (0.63) EGFRLRRK2
SCHEMBL5021150 0.76 LRRK2 (0.46) EGFRLRRK2ALKINSR
SCHEMBL4542112 0.75 LRRK2 (0.52) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed