SCHEMBL5021150

SCHEMBL5021150

COc1nc(Nc2cnn(C(C)(C)N)c2C)ncc1Cl

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 15/20 0.46
EGFR P00533 3/20 0.38
MAPK1 P28482 1/20 0.35
INSR P06213 1/20 0.35
ALK Q9UM73 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18426068 0.90 LRRK2 (0.47) LRRK2MAPK1INSRALK
SCHEMBL4542329 0.85 LRRK2 (0.46) LRRK2EGFR
SCHEMBL4562363 0.85 LRRK2 (0.58) LRRK2
SCHEMBL4537127 0.81 LRRK2 (0.63) LRRK2EGFRMAPK1
SCHEMBL27939108 0.81 LRRK2 (0.43) LRRK2MAPK1
SCHEMBL4542112 0.78 LRRK2 (0.52) LRRK2
SCHEMBL5021149 0.78 LRRK2 (0.54) LRRK2
SCHEMBL5021172 0.76 EGFR (0.48) LRRK2EGFRINSRALK
SCHEMBL4531370 0.75 LRRK2 (0.58) LRRK2MAPK1INSRALK
SCHEMBL4538610 0.75 LRRK2 (0.47) LRRK2EGFRINSRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed