SCHEMBL5021772

SCHEMBL5021772

O=C1N[C@@H](c2cccc(Br)c2)CO1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.42
EPAS1 Q99814 5/20 0.41
KMT2A Q03164 3/20 0.41
POLB P06746 3/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP19A1 P11511 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30370014 1.00 KDM1A (0.42) KDM1AEPAS1KMT2APOLBMEN1
SCHEMBL28983102 1.00 KDM1A (0.42) KDM1AEPAS1KMT2APOLBMEN1
SCHEMBL30370299 1.00 KDM1A (0.42) KDM1AEPAS1KMT2APOLBMEN1
SCHEMBL28983100 1.00 KDM1A (0.42) KDM1AEPAS1KMT2APOLBMEN1
SCHEMBL28983074 0.82 CYP19A1 (0.47) KMT2ACYP19A1KDM4EL3MBTL1
SCHEMBL31494783 0.82 CYP19A1 (0.47) KMT2AMEN1CYP19A1KDM4ENPC1
SCHEMBL30370012 0.82 CYP19A1 (0.47) KMT2ACYP19A1KDM4EL3MBTL1
SCHEMBL1439397 0.82 SLC6A3 (0.48) EPAS1KMT2AMEN1CYP19A1ALDH1A1
SCHEMBL30370325 0.82 CYP19A1 (0.47) KMT2AMEN1CYP19A1KDM4ENPC1
SCHEMBL28983054 0.82 SLC6A3 (0.48) EPAS1KMT2AMEN1CYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064603-A1 OXAZOLIDINONES AS MODULATORS OF MGLUR5 BRISTOL-MYERS SQUIBB COMPANY (US) 2012-05-18 WO disclosed