SCHEMBL5024294

SCHEMBL5024294

O[C@H]1[C@@H]2CC[C@H]1CNC2

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1726764 1.00
SCHEMBL5024292 1.00
SCHEMBL12153077 1.00
Hydrochloric Acid SCHEMBL6773968 0.97 CCR5 (0.47)
Hydrochloric Acid SCHEMBL6773969 0.97 CCR5 (0.47)
SCHEMBL16637274 0.88 CCR5 (0.44)
SCHEMBL30539390 0.88 CCR5 (0.44)
Hydrochloric Acid SCHEMBL6777912 0.85 CCR5 (0.42)
Hydrochloric Acid SCHEMBL6777914 0.85 CCR5 (0.42)
SCHEMBL21561562 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10189836-B2 Therapeutic compounds, compositions and methods of use thereof GENENTECH, INC. (US) 2019-01-29 US disclosed
EP-3390402-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF H. Hoffnabb-La Roche Ag (CH) 2018-10-24 EP disclosed
US-20180297997-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2018-10-18 US disclosed
WO-2017103188-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-06-22 WO disclosed
WO-2008044702-A1 PROCESS FOR PRODUCTION OF AZABICYCLOALKANOL DERIVATIVE NIPPON SODA CO., LTD. (JP) 2008-04-17 WO disclosed