4-Aminoquinazoline

4-Aminoquinazoline

SCHEMBL5026560

Nc1ncnc2ccccc12.O=C(O)C(F)(F)F

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 2/20 0.68
PI4K2B Q8TCG2 2/20 0.68
PI4K2A Q9BTU6 2/20 0.68
PI4KB Q9UBF8 2/20 0.68
MAP4K4 O95819 9/20 0.47
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.42
LMNA P02545 1/20 0.41
DCPS Q96C86 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
BCAT2 O15382 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Aminoquinazoline SCHEMBL29481714 1.00 PI4KA (0.68) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL28258394 0.86 PI4KA (0.78) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL28258393 0.86 PI4KA (0.78) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL27977310 0.84 PI4KA (0.81) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL28181385 0.84 PI4KA (0.95) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL142513 0.82 PI4KA (1.00) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL31377585 0.82 PI4KA (1.00) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL29363315 0.82 PI4KA (1.00) PI4KAPI4K2BPI4K2API4KBMAP4K4
4-Aminoquinazoline SCHEMBL28259933 0.82 PI4KA (0.70) PI4KAPI4K2BPI4K2API4KBMAP4K4
Trifluoroacetic Acid SCHEMBL28853097 0.81 MAP4K4 (0.52) MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957462-A2 NOVEL 2-AMINO-HETEROCYCLES UDEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES Astra Zeneca AB (SE) 2008-08-20 EP claimed
WO-2007058583-A2 NOVEL 2-AMINO-HETEROCYCLES USEFUL IN THE TREATMENT OF ABETA-RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-05-24 WO claimed
CN-114269731-A KIF18A inhibitors 美国安进公司 2022-04-01 CN disclosed
CN-111763215-A Compound with nitrogen-containing heterocyclic structure and preparation method and application thereof 成都海博为药业有限公司 2020-10-13 CN disclosed
CN-1882572-A Quinazoline derivatives as antitumor agents ASTRAZENECA AB (SE) 2006-12-20 CN disclosed