SCHEMBL5027770

SCHEMBL5027770

CC(C)(C)OC(=O)Nc1ccc(F)c(Cl)c1.Nc1ccc(F)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.54
TSHR P16473 2/20 0.50
EGFR P00533 2/20 0.50
AURKB Q96GD4 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.49
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
MAPT P10636 3/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
LMNA P02545 1/20 0.49
SLC2A1 P11166 1/20 0.49
ALDH1A1 P00352 2/20 0.48
GAA P10253 1/20 0.48
FADS1 O60427 1/20 0.48
CASP3 P42574 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
RORC P51449 1/20 0.47
KDM4E B2RXH2 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3202901 0.92 HTT (0.62) HTTTSHREGFRAURKBSMN1; SMN2
SCHEMBL14600409 0.87 MEN1 (0.66) HTTTSHRSMN1; SMN2NPC1RAB9A
SCHEMBL14600412 0.84 HTT (0.60) HTTSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL1094945 0.81 CA12 (0.47) HTTALDH1A1GAARORC
SCHEMBL29448767 0.81 CA12 (0.47) HTTALDH1A1GAARORC
SCHEMBL12228592 0.81 AR (0.49) HTTTSHREGFRAURKBMAPT
SCHEMBL30668235 0.81 CA12 (0.47) HTTNPC1RAB9AMEN1KMT2A
SCHEMBL6814996 0.81 CA12 (0.47) HTTNPC1RAB9AMEN1KMT2A
SCHEMBL29666354 0.81 AR (0.49) HTTTSHREGFRAURKBMAPT
SCHEMBL23024750 0.80 MAP4K4 (0.49) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299381-B1 SUBSTITUTED QUINAZOLINE DERIVATIVES AND THEIR USE AS INHIBITORS ASTRAZENECA AB (SE) 2008-05-07 EP disclosed