SCHEMBL5031829

SCHEMBL5031829

C[CH]CC(O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.41
PDE2A O00408 1/20 0.37
CES2 O00748 1/20 0.35
TACR1 P25103 10/20 0.35
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31378991 0.81 PNMT (0.41) PNMTCES2TACR1
SCHEMBL15211541 0.81 PNMT (0.41) PNMTPDE2ACES2TACR1IDO1
SCHEMBL5610427 0.79 PDE2A (0.51) PNMTPDE2ACES2TACR1IDO1
SCHEMBL2394599 0.79 PDE2A (0.51) PNMTPDE2ACES2TACR1IDO1
SCHEMBL25920947 0.78 PNMT (0.47) PNMTPDE2ACES2TACR1IDO1
SCHEMBL6484095 0.76 PNMT (0.46) PNMTPDE2ACES2TACR1IDO1
SCHEMBL459815 0.76 PNMT (0.46) PNMTPDE2ACES2TACR1IDO1
SCHEMBL264592 0.76 PNMT (0.46) PNMTPDE2ACES2TACR1IDO1
SCHEMBL9903281 0.76 PNMT (0.42) PNMTPDE2ACES2TACR1
SCHEMBL17243750 0.75 PNMT (0.36) PNMTPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973546-B1 CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS MERCK SHARP & DOHME (US) 2012-06-13 EP disclosed
EP-1973546-A2 CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS Merck & Co., Inc. (US) 2008-10-01 EP disclosed
WO-2007081570-A2 CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS MERCK & CO., INC. (US) 2007-07-19 WO disclosed