SCHEMBL5032005

SCHEMBL5032005

NC(=O)Oc1ccccc1NC(=O)c1ccc(C(C(=O)Nc2ccccc2)C(=O)Nc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.68
HDAC3 O15379 5/20 0.68
HDAC2 Q92769 5/20 0.68
NCOR2 Q9Y618 4/20 0.48
NPC1 O15118 1/20 0.47
NR1I2 O75469 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
AHR P35869 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30091844 0.82 NPC1 (0.57) HDAC1HDAC3HDAC2NPC1NR1I2
SCHEMBL1754325 0.81 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR2
SCHEMBL1689265 0.81 HDAC1 (0.89) HDAC1HDAC3HDAC2NCOR2
SCHEMBL2108547 0.81 HDAC1 (0.76) HDAC1HDAC3HDAC2NCOR2
SCHEMBL1689210 0.79 HDAC1 (0.90) HDAC1HDAC3HDAC2NCOR2
SCHEMBL12506316 0.79 CACNA1B (0.57) HDAC1HDAC3HDAC2NCOR2NPC1
SCHEMBL5031017 0.78 HDAC1 (0.69) HDAC1HDAC3HDAC2NCOR2NPC1
SCHEMBL1689184 0.77 HDAC1 (0.90) HDAC1HDAC3HDAC2NCOR2
SCHEMBL1754078 0.76 HDAC1 (0.71) HDAC1HDAC3HDAC2NCOR2KMT2A
SCHEMBL1689223 0.76 HDAC1 (0.71) HDAC1HDAC3HDAC2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed