SCHEMBL5031017

SCHEMBL5031017

NC(=O)Oc1ccccc1NC(=O)c1ccc(C(F)(C(=O)Nc2ccccc2)C(=O)Nc2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.69
MLYCD O95822 1/20 0.47
HDAC3 O15379 2/20 0.47
NCOR2 Q9Y618 2/20 0.47
HDAC2 Q92769 1/20 0.47
KMT2A Q03164 3/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
NR1I2 O75469 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
AHR P35869 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
PTGS1 P23219 1/20 0.45
NAMPT P43490 1/20 0.44
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 2/20 0.43
SIRT2 Q8IXJ6 1/20 0.43
RXFP1 Q9HBX9 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1754073 0.82 HDAC1 (1.00) HDAC1HDAC3NCOR2HDAC2PTGS1
SCHEMBL2886460 0.81 HDAC1 (0.76) HDAC1HDAC3NCOR2HDAC2KMT2A
SCHEMBL30091844 0.81 NPC1 (0.57) HDAC1MLYCDHDAC3HDAC2KMT2A
SCHEMBL12506316 0.78 CACNA1B (0.57) HDAC1HDAC3NCOR2HDAC2KMT2A
SCHEMBL5032005 0.78 HDAC1 (0.68) HDAC1HDAC3NCOR2HDAC2KMT2A
SCHEMBL1753684 0.77 HDAC1 (0.65) HDAC1HDAC3NCOR2HDAC2KMT2A
SCHEMBL28901074 0.74 KMT2A (0.57) HDAC1MLYCDHDAC3NCOR2HDAC2
SCHEMBL28347463 0.74 KMT2A (0.53) HDAC1MLYCDHDAC3HDAC2KMT2A
SCHEMBL2108610 0.73 HDAC1 (0.63) HDAC1HDAC3NCOR2HDAC2NPC1
SCHEMBL28254575 0.73 KMT2A (0.56) HDAC1MLYCDHDAC3NCOR2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed